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| Synthesis of Novel 3-Aminoazetidine Derivatives |
| MAO Ze-wei， ZHANG Meng-di， RAO Gao-xiong |
| School of Pharmacy, Yunnan University of Traditional Chinese Medicine， Kunming 650500， China |
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Abstract 1-（4-Acetylphenyl)-3-hydroxyazetidine（1） was prepared by reaction of 3-hydroxyazetidine with 4-fluoroacetophenone. Six novel 3-aminoazetidine derivatives were synthesized by methanesulfonyl, substitution， reduction and acylation reaction from 1. The structures were characterized by 1H NMR and 13C NMR.
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Received: 02 December 2014
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2015, Vol. 23 
